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Enzymes

Enzymes are globular proteins that can act as a biological catalyst to speed up any particular chemical reaction, by lowering the activation energy, without altering themselves.

​Enzymes are known as biological catalysts due to the following reasons:

  • They are known as biological because they are protein in nature and can only be made by living cells.

  • They are known as catalysts as they speed up a particular chemical reaction.


The lock and key hypothesis

  • As all enzymes are globular proteins they have a precise 3-D shape and have a "dent" on them known as the active site.

  • The substrate molecules have a shape which is complementary to the active site.

  • The substrates can easily fit into it like a lock (enzyme) and key (substrate).

  • An enzyme-substrate complex is formed and the enzyme catalyses the reaction.


Induced fit hypothesis

  • The shape of the substrate is not exactly complementary to the active site shape.

  • The active site is partially flexible and changes its shape slightly when the substrate binds.

  • Enzyme substrate complex forms.

  • It lowers the activation energy so the products form.


Intracellular enzymes: Enzymes that are used in the cell after being produced inside the cell. Extracellular enzymes: Enzymes that are outside in the cell after being produced inside the cell.


Effect of temperature on enzyme-catalyzed reaction

  • Increasing temperature increases the rate of reaction.

  • At higher temperatures, the kinetic energy of the enzyme and substrate will be higher.

  • The frequency of collision between enzyme and substrate will increase.

  • More enzyme-substrate complexes are formed.


  • All enzymes work best at a particular temperature which is known as optimum temperature.

  • If the temperature increases beyond this the hydrogen bonds that hold the tertiary structure of the enzyme break.

  • The active site gets deformed and the enzyme becomes denatured.

  • Substrate molecules cannot fit so, no enzyme-substrate complex form.


Effect of pH on enzyme catalysed reaction

  • All enzymes work best at a particular pH known as optimum pH.

  • If pH becomes too low or too high the solution will contain more H+ or OH- ions.

  • The presence of these enzymes will alter and destroy the ionic bonds that hold up the tertiary structure.

  • The active site gets deformed and the enzyme becomes denatured.

  • Substrate molecules cannot fit so, no enzyme-substrate complex form.



Effect of substrate concentration on enzyme catalysed reaction



  • As substrate concentration increases the initial rate of reaction increases up to a certain limit.

  • At this point all the substrate molecules are occupying enzymes active site, the enzymes are in excess.

  • Fixed amount of substrate is limiting the rate.


Enzyme Inhibitors

  • It is a substance that reduces the rate of enzyme-controlled reaction by combing with the enzyme.


Competitive Inhibitor :

  • A molecule that has a shape similar to the substrate.

  • It fits the active site instead of the substrate.

  • Enzyme inhibitor-complex is formed.

  • The substrate molecules can no longer fit the active site.

  • Fewer enzyme-substrate complex forms so fewer products form.


Non-Competitive inhibitor:

  • A molecule that attaches to the enzymes allosteric site.

  • The tertiary structure of the enzyme gets distorted.

  • The shape of the active site changes.

  • Substrate molecules are no longer complementary.

  • They do this by inducing polarity.



The Michaelis–Menten constant Km.

It is the concentration of the substrate to reach half of the Vmax . Km shows the affinity of enzyme for its substrate. A higher value of Km indicates a lower affinity for its substrate.


  • To calculate the Km of any enzyme first find the Vmax.

  • Then find half of the Vmax.

  • Read the substrate concentration from the x-axis to reach half the Vmax.



  • Enzyme A has the lowest Km so it has the highest affinity for its substrate.

  • Enzyme B has the lowest affinity as it has the highest (x-axis) Km value.



  • Inhibitor A is a competitive inhibitor.

  • It does not alter the Km of the reaction.

  • Some substrates can always bind to form a product so the reaction does reach Vmax.

  • But more substrate is required to do this.

  • Therefore the Km value of the enzyme increases.

  • Increasing the substrate concentration decreases the effect of competitive inhibitors.


  • Inhibitor B is a non-competitive inhibitor.

  • It binds to the allosteric site so it does not alter the affinity, therefore Km value remains the same.

  • It does decrease the Vmax of the reaction as all the enzymes are not active in the presence of a non-competitive inhibitor.


Immobilising Enzymes


Process:​

  • The enzyme to be immobilised is mixed with a solution of sodium alginate.

  • This mixture is dripped through a syringe into a solution of calcium chloride.

  • The calcium ions displace sodium ions forming NaCl & Calcium Alginate beads.

  • Calcium Alginate is hard and insoluble with the enzyme trapped in it.

  • The beads are left to harden further.


Advantages:

  • The product formed will have no enzymes so no purification steps are needed.

  • The enzymes can be reused.

  • Immobilised enzymes are more tolerant to temperature & pH changes





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